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Synthetic Heterocycles

702 Words3 Pages

1.Introduction: Ox diazole, a heterocycles nucleus has attracted a wide attention of the chemist in search for new therapeutic molecules.Five member heterocycles compounds show various type of biological activities among than 2,5-distributed 1,3,4-ox diazole are associated with diverse biological activities [2]. Various biological activities like antimicrobial, anti-tubercular, anti-inflammatory, Anticonvulsant [3], Hypnotic , Anesthetic activity [4]. 1,3,4-ox diazole showed antibacterial properties similar to those of well known sulfonamide drugs. The ox diazole nucleus with N=C-S linkage exhibits a large number of pharmacological activities [5]. Sulfone derivatives containing heterocycles moiety are known for their interesting …show more content…

The chemistry of heterocycles compounds is one of the most complex branches of chemistry. It is equally interesting for its theoretical implication for the diversity of its synthetic procedure and for the physiological and industrial significance. Synthetic heterocycles chemistry has influenced almost every place of human life and the heterocycles compounds have found their application in diverse fields medicine, agriculture, polymer, and various industries. Synthetic heterocycles drugs are used as Hypnotics, Anticonvulsants, Antiseptics, Antineoplastics, Antiviral, Antihistaminic, Anti-tumor etc. Majority of the large number of drugs being introduces in pharmacopeias every year are heterocycles …show more content…

The chemistry of heterocycles compounds is one of the most complexes of branches of chemistry. It is equally interesting for its theoretical implication for the diversity of its synthetic procedure and for the physiological and industrial significance. Synthetic heterocycles chemistry has influenced almost every place of human life and the heterocycles compounds have found their application in diverse field as medicine, agriculture, polymer, and various industries. The proposed work is in context with the compounds having 1,3,4-ox diazoles moiety. The other moieties like azetidinones, pyrrole and pyrolidines etc. also present and these moieties containing drugs have potential utility. Thus the combined molecules of 1,3,4-oxadiazoles and these heterocycles, it is expected that the novel heterocycles will have good antimicrobial properties and will be applied as

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